Multifaceted Telmisartan: Candidate for new therapeutic approaches

  • Prince Sanjeev Yoganand New Prince Hospital, GH South Care Street, Kadayanallur, Tirunelveli
  • Raison Chacko Dr. Raison P Chacko, Doctors Quarter, ESAF Hospital & Research Centre, Mannarkkad Road, Thachampara, Palakkad
  • Rajeshwar Kant Chandra Mishra Sanjeevni Clinic Gorakhpur
  • RLV Phani Kumar Sri Balaji Clinic and Diabetic Care, Bhavani Puram, Vijayawada
  • Saikat Kundu Diamond Harbour Road, Naiya Para, West Bengal
Keywords: PPAR γ, telmisartan, cardiovascular

Abstract

Telmisartan is an Angiotensin II type 1 (AT1) receptor blockers (ARBs), that is highly selective for the AT1 receptor and has a long duration of action because of its long terminal elimination half-life1. Telmisartan is considered to be the most potent member of the sartan group because, in addition to AT1R blockade, it strongly activates the antiinflammatory nuclear receptor, peroxisome proliferator-activated receptor γ (PPAR γ)

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References

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How to Cite
1.
Prince Sanjeev Yoganand, Raison Chacko, Rajeshwar Kant Chandra Mishra, RLV Phani Kumar, Saikat Kundu. Multifaceted Telmisartan: Candidate for new therapeutic approaches. Med. res. chronicles [Internet]. 1 [cited 2024Dec.22];7(1):45-9. Available from: https://medrech.com/index.php/medrech/article/view/416
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Original Research Article